SCHEMBL30006849

SCHEMBL30006849

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(F)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C(F)(F)F)nnc12

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.39
IRAK4 Q9NWZ3 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
MAPT P10636 1/20 0.32
CNR2 P34972 2/20 0.32
ADCY8 P40145 1/20 0.32
ADCY1 Q08828 1/20 0.32
RIPK1 Q13546 2/20 0.31
EPHX2 P34913 2/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
ACHE P22303 1/20 0.31
POLB P06746 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28909219 1.00 CFTR (0.39) CFTRIRAK4HCRTR1HCRTR2MAPT
SCHEMBL25687424 1.00 CFTR (0.39) CFTRIRAK4HCRTR1HCRTR2MAPT
SCHEMBL23958644 0.92 CFTR (0.36) CFTRMAPTCNR2ROCK2ROCK1
SCHEMBL30007924 0.92 CFTR (0.36) CFTRMAPTCNR2ROCK2ROCK1
SCHEMBL23958706 0.92 CFTR (0.36) CFTRMAPTCNR2ROCK2ROCK1
SCHEMBL25687411 0.92 CFTR (0.36) CFTRMAPTCNR2ROCK2ROCK1
SCHEMBL23958761 0.91 CFTR (0.35) CFTRIRAK4MAPTCNR2RIPK1
SCHEMBL23958708 0.91 CFTR (0.35) CFTRIRAK4MAPTCNR2RIPK1
SCHEMBL30007745 0.90 CFTR (0.34) CFTRMAPTCNR2RIPK1ROCK2
SCHEMBL25686209 0.90 CFTR (0.34) CFTRMAPTCNR2RIPK1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed