SCHEMBL30007214

SCHEMBL30007214

COc1cc(C(=O)NCC(O)(c2nc(-c3ccc(F)cc3)c(F)c(C(C)(C)O)c2F)C(F)(F)F)cc2cc(C3CC3)cnc12

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.35
GABRA5 P31644 4/20 0.33
CNR2 P34972 1/20 0.32
RIPK1 Q13546 2/20 0.32
PDE4B Q07343 2/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
MAPT P10636 1/20 0.31
ULK1 O75385 1/20 0.31
NR3C1 P04150 1/20 0.31
HPGDS O60760 1/20 0.30
JAK2 O60674 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28960598 1.00 CFTR (0.35) CFTRGABRA5CNR2RIPK1PDE4B
SCHEMBL25687302 1.00 CFTR (0.35) CFTRGABRA5CNR2RIPK1PDE4B
SCHEMBL30007175 0.89 CFTR (0.37) CFTRGABRA5RIPK1MAPTULK1
SCHEMBL25240950 0.89 CFTR (0.37) CFTRGABRA5RIPK1MAPTULK1
SCHEMBL25686191 0.89 CFTR (0.37) CFTRGABRA5RIPK1MAPTULK1
SCHEMBL25687494 0.87 CFTR (0.37) CFTRGABRA5CNR2RIPK1PDE4B
SCHEMBL25234891 0.87 CFTR (0.36) CFTRGABRA5CNR2ROCK2ROCK1
SCHEMBL30007228 0.86 CFTR (0.38) CFTRGABRA5CNR2MAPTNR3C1
SCHEMBL25235693 0.86 CFTR (0.38) CFTRGABRA5CNR2MAPTNR3C1
SCHEMBL25686201 0.86 CFTR (0.38) CFTRGABRA5CNR2MAPTNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed