SCHEMBL30007790

SCHEMBL30007790

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C(F)(F)F)cc2cc(C)cnc12

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CFTR P13569 5/20 0.38
NR3C1 P04150 1/20 0.34
GABRA5 P31644 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ULK1 O75385 1/20 0.33
PTGFR P43088 2/20 0.33
CNR2 P34972 1/20 0.33
RIPK1 Q13546 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25687207 1.00 CFTR (0.38) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL25280846 1.00 CFTR (0.38) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL25687495 0.93 CFTR (0.39) CFTRNR3C1GABRA5ALDH1A1NPSR1
SCHEMBL25687501 0.92 CFTR (0.39) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL23958707 0.91 CFTR (0.39) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL25687310 0.91 CFTR (0.39) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL25687266 0.91 CFTR (0.34) CFTRGABRA5ULK1
SCHEMBL25280037 0.91 CFTR (0.34) CFTRGABRA5ULK1
SCHEMBL25687500 0.91 CFTR (0.36) CFTRNR3C1GABRA5KDM4EALDH1A1
SCHEMBL23958734 0.89 CFTR (0.38) CFTRNR3C1GABRA5KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed