SCHEMBL30007990

SCHEMBL30007990

CC1(C)C=C(OS(=O)(=O)C(F)(F)F)c2cccnc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
CHRM1 P11229 1/20 0.32
PTGS2 P35354 3/20 0.32
KEAP1 Q14145 1/20 0.31
TDP2 O95551 1/20 0.30
NSD2 O96028 1/20 0.30
ABL1 P00519 1/20 0.30
PLCG1 P19174 1/20 0.30
CES1 P23141 1/20 0.30
PAX8 Q06710 1/20 0.30
RIN1 Q13671 1/20 0.30
MEN1 O00255 1/20 0.30
THRB P10828 1/20 0.30
BLM P54132 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
GAA P10253 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29060307 1.00 PDE4A (0.34) PDE4APDE4CPDE4DCHRM1PTGS2
SCHEMBL25717148 0.77 CHRM1 (0.34) CHRM1
SCHEMBL29060206 0.70
SCHEMBL30007549 0.70
SCHEMBL315126 0.70 PDE4A (0.40) PDE4APDE4CPDE4D
SCHEMBL21260401 0.69 PDE4A (0.39) PDE4APDE4CPDE4DPTGS2PTGS1
SCHEMBL14162088 0.69 CHRM1 (0.35) CHRM1
SCHEMBL16381650 0.68 PDK2 (0.31)
SCHEMBL15635309 0.68 PDK2 (0.35) PDE4APDE4CPDE4D
SCHEMBL3859888 0.68 CYP19A1 (0.37) PDE4APDE4CPDE4DTDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237825-A1 AZAARYL DERIVATIVE WITH EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-11-17 WO disclosed