SCHEMBL30008079

SCHEMBL30008079

C[C@H](Nc1cc(Cl)nc2c1cnn2[C@@H]1O[C@H](CO)[C@H]2OC(C)(C)O[C@H]21)c1ccccc1F

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NT5E P21589 12/20 0.59
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
SCN1A P35498 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22104979 1.00 NT5E (0.59) NT5EADORA2AADORA2BPI4KAPI4K2B
SCHEMBL27206558 1.00 NT5E (0.59) NT5EADORA2AADORA2BPI4KAPI4K2B
SCHEMBL30007724 0.87 NT5E (0.65) NT5E
SCHEMBL27206798 0.87 NT5E (0.65) NT5E
SCHEMBL24672775 0.87 NT5E (0.65) NT5E
SCHEMBL27195208 0.87 NT5E (0.62) NT5E
SCHEMBL24672776 0.86 NT5E (0.60) NT5E
SCHEMBL24672309 0.86 NT5E (0.73) NT5EADORA2AADORA2B
SCHEMBL22104978 0.86 NT5E (0.73) NT5EADORA2AADORA2B
SCHEMBL30008475 0.86 NT5E (0.73) NT5EADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4353732-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF Xizang Haisco Pharmaceutical Co., Ltd. (CN) 2024-04-17 EP disclosed
WO-2022237747-A1 SMALL MOLECULAR CD73 ANTAGONIST AND USE THEREOF 四川海思科制药有限公司 2022-11-17 WO disclosed