SCHEMBL30009410

SCHEMBL30009410

O=C1COc2ccc(Nc3nc(Nc4cccc(O)c4)ncc3F)cc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SYK P43405 17/20 1.00
JAK1 P23458 1/20 0.60
JAK3 P52333 1/20 0.60
AURKA O14965 3/20 0.54
MAPK8 P45983 1/20 0.54
AURKB Q96GD4 1/20 0.54
CDK19 Q9BWU1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL656578 1.00 SYK (1.00) SYKJAK1JAK3AURKAMAPK8
SCHEMBL30009889 1.00 SYK (1.00) SYKJAK1JAK3AURKAMAPK8
SCHEMBL656760 1.00 SYK (1.00) SYKJAK1JAK3AURKAMAPK8
SCHEMBL657850 0.93 SYK (0.86) SYKJAK1JAK3AURKAMAPK8
SCHEMBL656397 0.93 SYK (0.86) SYKJAK1JAK3AURKAMAPK8
SCHEMBL656700 0.90 SYK (0.81) SYKAURKAMAPK8AURKBCDK19
SCHEMBL657167 0.86 SYK (0.75) SYKJAK1JAK3
SCHEMBL13007743 0.84 SYK (0.72) SYKJAK1JAK3AURKAMAPK8
SCHEMBL12854318 0.84 SYK (0.72) SYKJAK1JAK3
SCHEMBL2745738 0.84 SYK (0.72) SYKJAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041259-A1 FEEDER-BASED AND FEEDER-FREE STEM CELL CULTURE SYSTEMS FOR STRATIFIED EPITHELIAL STEM CELLS, AND USES RELATED THERETO University of Houston System (US) 2022-08-17 EP disclosed