SCHEMBL30037477

SCHEMBL30037477

CC[C@@H](c1cn(-c2ccc(F)cc2)nn1)n1cc(-c2cncnc2OC)c2c(N)ncnc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFTR P13569 9/20 0.46
SRC P12931 3/20 0.36
ALK Q9UM73 1/20 0.34
EGFR P00533 2/20 0.33
KDR P35968 3/20 0.32
TEK Q02763 3/20 0.32
CYP17A1 P05093 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP11B1 P15538 1/20 0.32
AXL P30530 1/20 0.32
ABL1 P00519 1/20 0.32
ABL2 P42684 1/20 0.32
LCK P06239 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162713 1.00 CFTR (0.46) CFTRSRCALKEGFRKDR
SCHEMBL20162784 1.00 CFTR (0.46) CFTRSRCALKEGFRKDR
SCHEMBL20162716 0.92 CFTR (0.50) CFTRSRCEGFRKDRTEK
SCHEMBL20162712 0.92 CFTR (0.50) CFTRSRCEGFRKDRTEK
SCHEMBL30538085 0.92 CFTR (0.50) CFTRSRCEGFRKDRTEK
SCHEMBL20162672 0.91 CFTR (0.48) CFTRSRCEGFRKDRABL1
SCHEMBL30036376 0.91 CFTR (0.48) CFTRSRCEGFRKDRABL1
SCHEMBL30538049 0.91 CFTR (0.48) CFTRSRCEGFRKDRABL1
SCHEMBL20162670 0.91 CFTR (0.48) CFTRSRCEGFRKDRABL1
SCHEMBL20162643 0.89 CFTR (0.52) CFTRSRCALKCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115850268-A Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2023-03-28 CN claimed
CN-115850268-A Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2023-03-28 CN disclosed
CN-110337294-B Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2022-11-01 CN disclosed