SCHEMBL30037576

SCHEMBL30037576

CC[C@@H](c1cn(-c2ccccc2F)nn1)n1cc(C2CC2)c2c(N)ncnc21

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CFTR P13569 14/20 0.56
SRC P12931 2/20 0.37
PIK3CD O00329 1/20 0.36
NOTUM Q6P988 1/20 0.36
PI4KA P42356 1/20 0.34
PI4K2B Q8TCG2 1/20 0.34
PI4K2A Q9BTU6 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
METTL3 Q86U44 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162641 1.00 CFTR (0.56) CFTRSRCPIK3CDNOTUMPI4KA
SCHEMBL30538081 1.00 CFTR (0.56) CFTRSRCPIK3CDNOTUMPI4KA
SCHEMBL20162639 1.00 CFTR (0.56) CFTRSRCPIK3CDNOTUMPI4KA
SCHEMBL30038273 0.88 CFTR (0.46) CFTRNOTUMPI4KAPI4K2BPI4K2A
SCHEMBL30538114 0.88 CFTR (0.46) CFTRNOTUMPI4KAPI4K2BPI4K2A
SCHEMBL20162612 0.88 CFTR (0.46) CFTRNOTUMPI4KAPI4K2BPI4K2A
SCHEMBL20162611 0.88 CFTR (0.46) CFTRNOTUMPI4KAPI4K2BPI4K2A
SCHEMBL20162728 0.85 CFTR (0.59) CFTRSRCNOTUMPI4KAPI4K2B
SCHEMBL30036823 0.85 CFTR (0.59) CFTRSRCNOTUMPI4KAPI4K2B
SCHEMBL20162622 0.85 CFTR (0.45) CFTRSRCNOTUMPI4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115850268-A Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2023-03-28 CN claimed
CN-115850268-A Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2023-03-28 CN disclosed
CN-110337294-B Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会 2022-11-01 CN disclosed