SCHEMBL30043816

SCHEMBL30043816

CCn1ncc2cc(-c3ccc(C=O)cc3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.39
CACNA1H O95180 3/20 0.37
PTGER4 P35408 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ALDH3A1 P30838 1/20 0.37
ALDH1A3 P47895 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
TGFBR1 P36897 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMO O15229 1/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
RAD51 Q06609 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23497968 1.00 MCHR1 (0.39) MCHR1CACNA1HPTGER4ALDH1A1ALDH3A1
SCHEMBL3436601 0.88 CYP2A6 (0.46) CACNA1HPTGER4ALDH1A1ALDH3A1ALDH1A3
SCHEMBL21998159 0.81 BRD4 (0.45) MCHR1CYP3A4CYP2C19
SCHEMBL22926448 0.80 BRD4 (0.44) MCHR1CYP3A4CYP2C19
SCHEMBL27308857 0.79 CYP2A6 (0.46) PTGER4ALDH1A3HTR2AHTR2CCYP2A6
SCHEMBL22926449 0.78 BRD4 (0.36) MCHR1ALDH1A1ALDH1A3CYP3A4CYP2C19
SCHEMBL30044048 0.77 CYP2A6 (0.47) CACNA1HPTGER4HTR2AHTR2CCYP2A6
SCHEMBL23497966 0.77 CYP2A6 (0.47) CACNA1HPTGER4HTR2AHTR2CCYP2A6
SCHEMBL23511034 0.76 MAOB (0.39) CACNA1HHTR2AHTR2CKMO
SCHEMBL23807111 0.75 BRD4 (0.42) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4073054-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF TUMORS Fondazione Istituto Italiano di Tecnologia (IT) 2022-10-19 EP disclosed