SCHEMBL30085580

SCHEMBL30085580

Clc1ccc(-c2cc(N3CCN(c4ccccc4)CC3)nc(-c3cccnc3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.53
MAPT P10636 4/20 0.52
TSHR P16473 3/20 0.52
HSD17B10 Q99714 3/20 0.52
MAPK1 P28482 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
PIK3CB P42338 2/20 0.52
PIK3CG P48736 2/20 0.52
KDM4E B2RXH2 2/20 0.51
LMNA P02545 2/20 0.51
HPGD P15428 1/20 0.51
CYP3A4 P08684 6/20 0.49
CYP2C9 P11712 4/20 0.48
CYP2C19 P33261 4/20 0.48
CYP2D6 P10635 4/20 0.48
CYP1A2 P05177 3/20 0.48
RXFP1 Q9HBX9 1/20 0.48
CETP P11597 1/20 0.46
HRH4 Q9H3N8 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28894673 1.00 PIK3CA (0.53) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL30085611 0.91 PIK3CA (0.52) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL28894946 0.91 PIK3CA (0.52) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL28895016 0.90 PIK3CA (0.50) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL30085461 0.90 PIK3CA (0.50) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL30085378 0.90 MAPT (0.52) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL28894764 0.90 MAPT (0.52) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL28894548 0.88 PIK3CA (0.48) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL30085624 0.88 HPGD (0.59) PIK3CAMAPTTSHRHSD17B10MAPK1
SCHEMBL28894859 0.88 HPGD (0.59) PIK3CAMAPTTSHRHSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN claimed
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed