SCHEMBL30091654

SCHEMBL30091654

COc1ccc(Br)cc1-c1ccnc(N)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 5/20 0.52
MGAM O43451 1/20 0.50
GAA P10253 1/20 0.50
SI P14410 1/20 0.50
MGAM2 Q2M2H8 1/20 0.50
GSK3B P49841 1/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
NPC1 O15118 1/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
PPARG P37231 1/20 0.43
GFER P55789 1/20 0.43
NCOA2 Q15596 1/20 0.43
NCOA1 Q15788 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22272596 1.00 DYRK1A (0.52) DYRK1AMGAMGAASIMGAM2
SCHEMBL3361169 0.80 DYRK1A (0.60) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL320181 0.78 DYRK1A (0.54) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL23927489 0.77 DYRK1A (0.48) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL30091458 0.77 DYRK1A (0.48) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL6496645 0.76 GAA (0.51) MGAMGAASIMGAM2NPC1
SCHEMBL31381034 0.76 DYRK1A (0.73) DYRK1AGSK3BNOS3NOS1NOS2
SCHEMBL16371252 0.75 DYRK1A (0.55) DYRK1AGAAGSK3BNOS3NOS1
SCHEMBL4215294 0.75 CDK5 (0.52) DYRK1AMGAMGAASIMGAM2
SCHEMBL14125145 0.74 GAA (0.56) MGAMGAASIMGAM2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166116-B Amido bridged heterocyclic compound, and composition and application thereof 北京赛特明强医药科技有限公司 2022-12-27 CN disclosed