SCHEMBL30097237

SCHEMBL30097237

Nc1c[nH]c2c(NCc3ccc(B(O)O)cc3)ncnc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT1 Q99873 1/20 0.41
EGFR P00533 2/20 0.41
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CDK2 P24941 1/20 0.40
AURKA O14965 8/20 0.40
RPS6KB1 P23443 7/20 0.40
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
OXTR P30559 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
JAK2 O60674 2/20 0.38
JAK1 P23458 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27410555 1.00 PRMT1 (0.41) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL27409830 0.85 RPS6KB1 (0.48) AURKARPS6KB1AURKB
SCHEMBL30097217 0.85 RPS6KB1 (0.48) AURKARPS6KB1AURKB
SCHEMBL27409232 0.83 PRMT1 (0.39) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL30097224 0.82 EGFR (0.42) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL27410545 0.82 EGFR (0.42) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL27409290 0.81 AURKA (0.40) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL30097159 0.81 AURKA (0.40) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL27409242 0.81 AURKA (0.40) PRMT1EGFRMAPK1LMNACYP1A2
SCHEMBL30097205 0.80 PRMT1 (0.38) PRMT1EGFRMAPK1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022197734-A1 BICYCLIC HETEROARYL BORONATE DERIVATIVES AS ECTONUCLEOTIDE PYROPHOSPHATASE PHOSPHODIESTERASE 1 INHIBITORS RIBOSCIENCE LLC (US) 2022-09-22 WO disclosed