SCHEMBL30101807

SCHEMBL30101807

N#Cc1c(Cl)c2nc(Cl)ccc2[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 5/20 0.42
KDM4E B2RXH2 1/20 0.39
KDM5A P29375 1/20 0.38
KDM5C P41229 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
PDE2A O00408 1/20 0.37
PSMB8 P28062 1/20 0.36
XDH P47989 1/20 0.36
IDH1 O75874 3/20 0.36
KCNMA1 Q12791 1/20 0.36
PARP1 P09874 1/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22275062 1.00 PDE9A (0.42) PDE9AKDM4EKDM5AKDM5CKDM5B
SCHEMBL25389897 0.85 KDM5A (0.49) PDE9AKDM5AKDM5CKDM5BLMNA
SCHEMBL31298163 0.82 KDM5A (0.43) PDE9AKDM5AKDM5CKDM5BLMNA
SCHEMBL4754780 0.80 PDE9A (0.60) PDE9AKDM4EKDM5AKDM5CKDM5B
SCHEMBL22275250 0.74 PDE9A (0.64) PDE9A
SCHEMBL20870664 0.72 PDE9A (0.60) PDE9AKDM4EKDM5AKDM5CKDM5B
SCHEMBL22275077 0.71 PDE9A (0.65) PDE9A
SCHEMBL21840104 0.71 KDM4E (0.38) PDE9AKDM4ELMNAHPGDALDH1A1
SCHEMBL1790858 0.69 KDM4E (0.41) KDM4ELMNAALDH1A1CYP1A2PDE2A
SCHEMBL1621734 0.69 PDE9A (0.62) PDE9AKDM4ELMNAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111471059-B PDE9 inhibitors and uses thereof 药捷安康(南京)科技股份有限公司 2022-12-02 CN disclosed