Balamapimod

Balamapimod

SCHEMBL30104249

COc1cc2c(Nc3ccc(Sc4nccn4C)c(Cl)c3)c(C#N)cnc2cc1N1CCC(N2CCCC2)CC1

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

MAP2K1MAP2K2

The experimentally established mechanism targets of Balamapimod. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP2K1 known ✓ Q02750 13/20 0.73
IGF1R P08069 9/20 0.81
MAPK3 P27361 1/20 0.67
MAPK1 P28482 1/20 0.67
MAP3K1 Q13233 1/20 0.67
EGFR P00533 1/20 0.58
ERBB2 P04626 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Balamapimod SCHEMBL2965207 1.00 IGF1R (0.81) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2974425 0.99 IGF1R (0.80) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2963305 0.95 IGF1R (0.87) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2968693 0.94 IGF1R (0.78) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2962949 0.94 IGF1R (0.87) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2976171 0.94 IGF1R (0.71) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2975567 0.94 MAP2K1 (0.75) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL14418379 0.91 IGF1R (0.67) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2964257 0.91 IGF1R (0.82) IGF1RMAP2K1MAPK3MAPK1MAP3K1
SCHEMBL2966483 0.91 IGF1R (0.66) IGF1RMAP2K1MAPK3MAPK1MAP3K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250281607-A1 MEDICAMENT FOR TREATMENT AND/OR PREVENTION OF CANCER TORAY INDUSTRIES, INC. (JP) 2025-09-11 US disclosed
EP-4378478-A1 MEDICAMENT FOR TREATMENT AND/OR PREVENTION OF CANCER Toray Industries, Inc. (JP) 2024-06-05 EP disclosed
CN-117677398-A Medicine for treating and/or preventing cancer 东丽株式会社 2024-03-08 CN disclosed
WO-2023008462-A1 MEDICAMENT FOR TREATMENT AND/OR PREVENTION OF CANCER 東レ株式会社 2023-02-02 WO disclosed