SCHEMBL30104796

SCHEMBL30104796

FC(F)(F)c1ccc2c(c1)cc1n2CCNC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 11/20 0.62
HTR2A P28223 9/20 0.62
HTR1D P28221 2/20 0.41
ADRB1 P08588 2/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ADRB2 P07550 1/20 0.36
NCF1 P14598 1/20 0.36
KCNH2 Q12809 1/20 0.35
HTR2B P41595 1/20 0.34
IDH2 P48735 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13208414 0.85 HTR2A (0.62) HTR2CHTR2AHTR3AKCNH2
SCHEMBL4705406 0.80 HTR2A (0.68) HTR2CHTR2ASIGMAR1KCNH2
SCHEMBL3155248 0.79 HTR2C (0.69) HTR2CHTR2AKCNH2
SCHEMBL5917403 0.77 HTR2A (0.68) HTR2CHTR2AMAPT
SCHEMBL4705400 0.77 HTR2A (0.68) HTR2CHTR2AADRB1SIGMAR1MEN1
SCHEMBL5917499 0.77 HTR2C (1.00) HTR2CHTR2AADRB1HTR3EHTR3B
SCHEMBL6714516 0.77 HTR2C (0.55) HTR2CHTR2AHTR1DADRB1HTR3E
Hydrochloric Acid SCHEMBL5917431 0.76 HTR2C (0.97) HTR2CHTR2AHTR3EHTR3BHTR3A
SCHEMBL2356686 0.74 HTR2A (1.00) HTR2CHTR2AHTR3EHTR3BHTR3A
SCHEMBL24640538 0.74 HTR2C (0.42) HTR2CHTR2AHTR1DADRB1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed
WO-2022247839-A1 PARP7 INHIBITOR 山东轩竹医药科技有限公司 2022-12-01 WO disclosed