SCHEMBL30105906

SCHEMBL30105906

COc1cccc2c(NC3CCC(C=O)CC3)ncnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 4/20 0.50
CYP1A2 P05177 4/20 0.50
CYP2D6 P10635 4/20 0.50
CLK4 Q9HAZ1 4/20 0.50
CYP2C19 P33261 3/20 0.50
CYP3A4 P08684 3/20 0.50
TSHR P16473 3/20 0.50
LMNA P02545 2/20 0.50
RPS6KB1 P23443 5/20 0.47
AURKA O14965 4/20 0.47
EGFR P00533 1/20 0.46
ALDH1A1 P00352 2/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
JAK2 O60674 5/20 0.44
JAK1 P23458 5/20 0.44
IRAK4 Q9NWZ3 1/20 0.44
HSD17B10 Q99714 2/20 0.43
PDE5A O76074 1/20 0.42
NSD2 O96028 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28926184 1.00 USP2 (0.50) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL29062077 0.93 USP2 (0.46) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL29062075 0.93 USP2 (0.46) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL30105969 0.93 USP2 (0.46) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL28926243 0.84 USP2 (0.44) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL30105970 0.83 USP2 (0.49) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL28926188 0.83 USP2 (0.49) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL28926246 0.82 USP2 (0.43) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL28926173 0.81 CYP1A2 (0.50) USP2CYP1A2CYP2D6CLK4CYP2C19
SCHEMBL30105914 0.81 CYP1A2 (0.50) USP2CYP1A2CYP2D6CLK4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115536696-B ENPP1 inhibitors 上海齐鲁制药研究中心有限公司 2023-07-14 CN disclosed
CN-115536696-A ENPP1 inhibitors 上海齐鲁制药研究中心有限公司 2022-12-30 CN disclosed