SCHEMBL30108181

SCHEMBL30108181

COc1cc(N2CC(N(C)C)C2)c(N)cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.61
EGFR P00533 14/20 0.59
IGF1R P08069 3/20 0.53
KCNH2 Q12809 3/20 0.53
INSR P06213 2/20 0.53
CDK2 P24941 4/20 0.47
CCNT1 O60563 3/20 0.47
CDK9 P50750 3/20 0.47
CCNA2 P20248 2/20 0.47
CDK7 P50613 2/20 0.47
CCNH P51946 2/20 0.47
CDK1 P06493 1/20 0.47
KDR P35968 1/20 0.47
MNAT1 P51948 1/20 0.47
JUN P05412 1/20 0.47
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
MAPK10 P53779 1/20 0.47
CCNK O75909 2/20 0.47
CDK12 Q9NYV4 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14663305 1.00 ALK (0.61) ALKEGFRIGF1RKCNH2INSR
SCHEMBL14718803 0.94 ALK (0.64) ALKEGFRIGF1RKCNH2INSR
SCHEMBL29974570 0.88 EGFR (0.74) ALKEGFRIGF1RKCNH2CDK2
SCHEMBL14663439 0.88 EGFR (0.74) ALKEGFRIGF1RKCNH2CDK2
SCHEMBL14663492 0.88 EGFR (0.57) ALKEGFRIGF1RKCNH2INSR
SCHEMBL30956860 0.87 ALK (0.68) ALKEGFRIGF1RKCNH2CDK2
SCHEMBL29232057 0.87 ALK (0.68) ALKEGFRIGF1RKCNH2CDK2
SCHEMBL14719276 0.86 EGFR (0.80) EGFRIGF1RKCNH2INSRCDK2
SCHEMBL30108177 0.85 FLT3 (0.60) EGFRIGF1RKCNH2CDK2CDK1
SCHEMBL14663301 0.85 FLT3 (0.60) EGFRIGF1RKCNH2CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115650974-B N- [5- (pyrimidine-2-amino) -2, 4-disubstituted phenyl ] -cis-pentadiene amide derivative and application thereof 天津大学 2024-06-18 CN disclosed
CN-115650974-A N- [5- (pyrimidine-2-amino) -2,4-disubstituted phenyl ] -cis-pentadiene amide derivative and application thereof 天津大学 2023-01-31 CN disclosed