SCHEMBL30114830

SCHEMBL30114830

COc1cccc(C)c1NC(=O)c1ccc(Nc2ncc(SC)c(-c3cccnc3F)n2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.42
ABL1 P00519 4/20 0.40
BCR P11274 4/20 0.40
IGF1R P08069 1/20 0.39
ABCB1 P08183 1/20 0.38
CHRNA7 P36544 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
AURKA O14965 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21799104 1.00 PTK2 (0.42) PTK2ABL1BCRIGF1RABCB1
SCHEMBL20188131 0.95 PTK2 (0.44) PTK2ABL1BCRABCB1LMNA
SCHEMBL30530287 0.95 PTK2 (0.44) PTK2ABL1BCRABCB1LMNA
SCHEMBL21799106 0.93
SCHEMBL20187976 0.89 AURKA (0.45) AURKA
SCHEMBL30114850 0.89 AURKA (0.45) AURKA
SCHEMBL20196486 0.86 AURKA (0.47) ABL1BCRLMNAMAPTAURKA
SCHEMBL30114870 0.86 AURKA (0.47) ABL1BCRLMNAMAPTAURKA
SCHEMBL21799064 0.86 ABL1 (0.39) PTK2ABL1BCRABCB1
SCHEMBL30114857 0.86 ABL1 (0.39) PTK2ABL1BCRABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139692-B Heteroaryl amine compounds for modulating hedgehog pathway and methods of making and using the same 财团法人生物技术开发中心 2023-08-25 CN disclosed
EP-3544685-B1 HETROARYLAMINE COMPOUNDS FOR MODULATING THE HEDGEHOG PATHWAY AND PREPARING METHOD AND USES THEREOF DEV CT BIOTECHNOLOGY (TW) 2023-01-04 EP disclosed