SCHEMBL30128063

SCHEMBL30128063

COc1ncc(-c2ccncc2)c2sc(NC(=O)c3ccc(C(=O)N(C)C)cc3)nc12

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 4/20 0.48
POLQ O75417 1/20 0.44
CSNK2A1 P68400 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
DUSP3 P51452 1/20 0.41
ADORA2A P29274 4/20 0.41
ADORA2B P29275 4/20 0.41
ADORA1 P30542 4/20 0.41
LMNA P02545 1/20 0.41
CLK1 P49759 1/20 0.41
CLK2 P49760 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20702376 1.00 CHRM4 (0.48) CHRM4POLQCSNK2A1SMN1; SMN2ALDH1A1
SCHEMBL20705299 0.91 CHRM4 (0.48) CHRM4POLQCSNK2A1SMN1; SMN2ALDH1A1
SCHEMBL30127887 0.91 CHRM4 (0.48) CHRM4POLQCSNK2A1SMN1; SMN2ALDH1A1
SCHEMBL20702388 0.91 CSNK2A1 (0.46) POLQCSNK2A1SMN1; SMN2ALDH1A1TP53
SCHEMBL22027634 0.85 ADORA2A (0.44) POLQCSNK2A1SMN1; SMN2ALDH1A1TP53
SCHEMBL30127873 0.85 ADORA2A (0.44) POLQCSNK2A1SMN1; SMN2ALDH1A1TP53
SCHEMBL24713254 0.82 ADORA1 (0.44) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL22063533 0.82 ADORA2A (0.50) CHRM4SMN1; SMN2ALDH1A1ADORA2AADORA2B
SCHEMBL20702441 0.82 POLQ (0.47) POLQCSNK2A1SMN1; SMN2ALDH1A1TP53
SCHEMBL20702421 0.81 ADORA1 (0.47) SMN1; SMN2ALDH1A1DUSP3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3661941-B1 THIAZOLOPYRIDINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2022-12-14 EP claimed