SCHEMBL301296

SCHEMBL301296

COc1cccc(P(c2ccccc2)c2ccccc2)c1-c1c(OC)cccc1P(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA7 P43166 3/20 0.44
CA9 Q16790 3/20 0.44
CA12 O43570 2/20 0.44
CA14 Q9ULX7 2/20 0.44
CA4 P22748 1/20 0.44
DRD1 P21728 2/20 0.41
TDP1 Q9NUW8 4/20 0.41
CYP3A4 P08684 2/20 0.41
TOP1 P11387 1/20 0.38
ALDH1A1 P00352 5/20 0.38
TP53 P04637 2/20 0.38
TSHR P16473 1/20 0.38
ADRA2B P18089 1/20 0.38
PTGS1 P23219 1/20 0.38
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29430119 1.00 CA1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL6565552 1.00 CA1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL29407955 1.00 CA1 (0.44) CA1CA2CA7CA9CA12
SCHEMBL1768301 0.98 CA1 (0.43) CA1CA2CA7CA9CA12
SCHEMBL13593792 0.92 CA1 (0.38) CA1CA2CA7CA9CA12
SCHEMBL12083834 0.92 CA12 (0.38) CA1CA2CA7CA9CA12
SCHEMBL7289398 0.90 CA1 (0.36) CA1CA2CA7CA9CA12
SCHEMBL5573142 0.90 CA1 (0.36) CA1CA2CA7CA9CA12
SCHEMBL5195630 0.90 APP (0.44) CA1CA2CA7CA9CA12
SCHEMBL1768406 0.90 TOP1 (0.41) CA1CA2CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 656 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3710422-B1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY AND DIASTEREOMERICALLY ENRICHED CYCLOBUTANE AMINES AND AMIDES SYNGENTA CROP PROTECTION AG (CH) 2026-01-07 EP claimed
CN-118206463-A Method for synthesizing tetrahydronaphthalene compounds through asymmetric hydrogenation of amide-guided naphthalene compounds 中国科学院大连化学物理研究所 2024-06-18 CN claimed
CN-117263897-A Chiral dibenzosubenol compound and asymmetric synthesis method thereof 四川师范大学 2023-12-22 CN claimed
CN-116947580-A Method for constructing axial chiral compound by hydrogenation and desymmetry of rhodium-catalyzed anthracene 中国科学院大连化学物理研究所 2023-10-27 CN claimed
CN-116410118-A Preparation method of beta-lactam compound 中国科学技术大学 2023-07-11 CN claimed
CN-114669333-B Catalyst system and catalytic method for catalyzing decarbonylation hydrogenation of alpha-quaternary carbon aldehyde 中山大学 2023-06-23 CN claimed
CN-113754889-B Method for synthesizing polysilicone through selective dehydrogenation coupling of polysilicone and cobalt-catalyzed latent chiral silane and diol 中国科学院大连化学物理研究所 2022-10-14 CN claimed
CN-114669333-A Catalyst system and method for catalyzing decarbonylation and hydrogenation of alpha-quaternary carbon aldehyde 中山大学 2022-06-28 CN claimed
EP-2964384-B1 AQUEOUS HYDROGENATION REACTIONS USING WATER-INSOLUBLE RUTHENIUM CATALYST COMPOSITION DUDECHEM GMBH (DE) 2022-05-04 EP claimed
CN-113754889-A Method for synthesizing polysilicone through selective dehydrogenation coupling of polysilicone and cobalt-catalyzed latent chiral silane and diol 中国科学院大连化学物理研究所 2021-12-07 CN claimed
US-6069245-A PRODUCING A 3-BENZOYLAMINO-4-BENZOYLOXYHEXAHYDROAZEPINE BY THE CATALYTIC HYDROGENATION OF THE 4-OXO-AMINE SALT DERIVATIVE; PROTECTING THE RING NITROGEN; FORMING A FUSED RING; HYDROLYSIS; ACYLATION AND DEPROTECTING HOFFMANN-LA ROCHE INC. (US) 2000-05-30 US claimed
EP-0974590-A1 Process for the preparation of chiral lactones by asymetrical hydrogenation F. HOFFMANN-LA ROCHE AG (CH) 2000-01-26 EP claimed
US-5902882-A ASYMMETRICALLY HYDROGENATING AN AZEPINE COMPOUND IN THE PRESENCE OF A RUTHENIUM-DIPHOSPHINE COMPLEX CATALYST HOFFMANN-LA ROCHE INC. (US) 1999-05-11 US claimed
US-5750690-A HYDROGENATION OF A 1,2-DIALKYLOXO-3-CARBOXY-3-PYRAZOLINE OR 1,2,5,6-TETRAHYDROPYRIDAZINE OR DERIVATIVE; INTERMEDIATES FOR THE HYPOTENSIVE AGENT, ?CILAZAPRIL? HOFFMANN-LA ROCHE INC. (US) 1998-05-12 US claimed
EP-0802190-A1 Process and intermediates for preparing azepines F. HOFFMANN-LA ROCHE AG (CH) 1997-10-22 EP claimed
US-5600015-A USING RUTHENIUM COMPLEX OF OPTICALLY ACTIVE ATROPISOMERIC DIPHOSPHINE LIGAND AS HYDROGENATION CATALYST HOFFMANN-LA ROCHE INC. (US) 1997-02-04 US claimed
US-5488172-A Chiral phosphorus compounds HOFFMANN-LA ROCHE INC. (US) 1996-01-30 US claimed
EP-0492401-B1 Asymmetric hydrogenation CIBA GEIGY AG (CH) 1996-01-24 EP claimed
EP-0398132-B1 Phosphorous compounds HOFFMANN LA ROCHE (CH) 1995-09-20 EP claimed
EP-0248800-B1 Process for making crosslinkable compositions BICC PLC (GB) 1995-08-23 EP claimed