SCHEMBL30137527

SCHEMBL30137527

Nc1nc(NCC2CCCNC2)cnc1Sc1cccc(Cl)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 13/20 0.50
CCNT1 O60563 7/20 0.45
KCNH2 Q12809 2/20 0.44
CDK9 P50750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30137522 0.94 PTPN11 (0.52) PTPN11CCNT1KCNH2
SCHEMBL25514421 0.89 CCNT1 (0.45) PTPN11CCNT1KCNH2CDK9
SCHEMBL30137467 0.89 PTPN11 (0.53) PTPN11CCNT1KCNH2
SCHEMBL30137518 0.86 PTPN11 (0.50) PTPN11CCNT1KCNH2
SCHEMBL19785342 0.83 PTPN11 (0.41) PTPN11CCNT1KCNH2CDK9
SCHEMBL30137526 0.83 PTPN11 (0.45) PTPN11KCNH2
SCHEMBL30137471 0.80 PTPN11 (0.49) PTPN11KCNH2
SCHEMBL30137457 0.77 PTPN11 (0.51) PTPN11CCNT1KCNH2
SCHEMBL25514397 0.77 PTPN11 (0.44) PTPN11CCNT1KCNH2
SCHEMBL19785567 0.77 PTPN11 (0.42) PTPN11CCNT1KCNH2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611869-A Heterocyclic pyrazine derivative and application thereof in preparation of SHP2 inhibitor 山东大学 2023-01-17 CN claimed
CN-115611869-B Heterocyclic pyrazine derivative and application thereof in preparation of SHP2 inhibitor 山东大学 2024-08-09 CN disclosed
CN-115611869-A Heterocyclic pyrazine derivative and application thereof in preparation of SHP2 inhibitor 山东大学 2023-01-17 CN disclosed