SCHEMBL30139732

SCHEMBL30139732

Cn1nc(N)c2cnc(N)nc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.50
GSK3B P49841 1/20 0.45
CDK4 P11802 1/20 0.43
CCND3 P30281 1/20 0.43
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
TLR9 Q9NR96 8/20 0.40
TLR8 Q9NR97 8/20 0.40
TLR7 Q9NYK1 8/20 0.39
PIK3CA P42336 1/20 0.36
MTOR P42345 1/20 0.36
RICTOR Q6R327 1/20 0.36
RPTOR Q8N122 1/20 0.36
MAPKAP1 Q9BPZ7 1/20 0.36
MLST8 Q9BVC4 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215554 0.83 CDK4 (0.42) BTKGSK3BCDK4CCND3TLR9
SCHEMBL4222561 0.81 CDK4 (0.41) BTKGSK3BCDK4CCND3PI4KA
SCHEMBL4233087 0.75 GRM5 (0.54) GSK3BPI4KBTLR9TLR8TLR7
SCHEMBL4227244 0.75 TLR7 (0.50) PI4KBTLR9TLR8TLR7PIK3CA
SCHEMBL4049229 0.75 ADORA2A (0.47) CDK4CCND3TLR9TLR8TLR7
SCHEMBL4218178 0.74 TLR7 (0.50) GSK3BCDK4CCND3TLR9TLR8
SCHEMBL4220294 0.74 TLR7 (0.47) BTKTLR9TLR8TLR7PIK3CA
SCHEMBL4215652 0.73 MTOR (0.39) GSK3BTLR9TLR8TLR7PIK3CA
SCHEMBL30861079 0.73 PI4KB (0.55) BTKGSK3BPI4KAPI4K2BPI4K2A
SCHEMBL27228218 0.73 PI4KB (0.55) BTKGSK3BPI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022270994-A1 NOVEL BIFUNCTIONAL HETEROCYCLIC COMPOUND HAVING BTK DEGRADATION FUNCTION VIA UBIQUITIN PROTEASOME PATHWAY, AND USE THEREOF 한국화학연구원 2022-12-29 WO disclosed