SCHEMBL30141355

SCHEMBL30141355

CS(=O)(=O)c1cc(NC(=O)c2c(C(F)(F)F)c(C3CC3)nn2CC2CCCCO2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 18/20 0.43
CNR2 P34972 1/20 0.37
MGAT2 Q10469 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24906447 1.00 SCN10A (0.43) SCN10ACNR2MGAT2
SCHEMBL24906475 1.00 SCN10A (0.43) SCN10ACNR2MGAT2
SCHEMBL24906303 0.98 SCN10A (0.43) SCN10ACNR2MGAT2
SCHEMBL30141416 0.88 SCN10A (0.44) SCN10A
SCHEMBL24757318 0.87 SCN10A (0.40) SCN10ACNR2
SCHEMBL30141451 0.87 SCN10A (0.40) SCN10ACNR2
SCHEMBL24758415 0.87 SCN10A (0.40) SCN10ACNR2
SCHEMBL24906422 0.87 SCN10A (0.44) SCN10A
SCHEMBL24906283 0.85 SCN10A (0.42) SCN10A
SCHEMBL24906223 0.85 SCN10A (0.42) SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4355733-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2024-04-24 EP claimed
WO-2022263498-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2022-12-22 WO claimed
EP-4355733-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2024-04-24 EP disclosed
WO-2022263498-A1 SUBSTITUTED PYRAZOLE AMIDES Grünenthal GmbH (DE) 2022-12-22 WO disclosed