SCHEMBL30153261

SCHEMBL30153261

Cn1nc(C(F)(F)F)cc1NC(=O)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 1/20 0.50
ORAI1 Q96D31 1/20 0.50
TRPV1 Q8NER1 1/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CRACR2A Q9BSW2 1/20 0.43
PTPN1 P18031 1/20 0.43
SLC6A3 Q01959 1/20 0.43
KCNH2 Q12809 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28398093 1.00 STIM1 (0.50) STIM1ORAI1TRPV1ALDH1A1CYP3A4
SCHEMBL28405257 0.90 STIM1 (0.48) STIM1ORAI1ALDH1A1CYP3A4HSD17B10
SCHEMBL30153355 0.90 STIM1 (0.48) STIM1ORAI1ALDH1A1CYP3A4HSD17B10
SCHEMBL28396543 0.89 STIM1 (0.53) STIM1ORAI1ALDH1A1RAB9A
SCHEMBL30153360 0.89 STIM1 (0.53) STIM1ORAI1ALDH1A1RAB9A
SCHEMBL28407309 0.87 STIM1 (0.44) STIM1ORAI1TRPV1ALDH1A1CYP3A4
SCHEMBL30153341 0.87 STIM1 (0.44) STIM1ORAI1TRPV1ALDH1A1CYP3A4
SCHEMBL28405278 0.87 STIM1 (0.46) STIM1ORAI1PTPN1BRAFFLT3
SCHEMBL30153384 0.87 STIM1 (0.46) STIM1ORAI1PTPN1BRAFFLT3
SCHEMBL31703953 0.86 LRRK2 (0.43) STIM1ORAI1TRPV1CRACR2APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111187215-B Fluorine-containing pyrazole amide derivative, preparation method and application thereof 西北农林科技大学 2023-02-24 CN disclosed