SCHEMBL30158950

SCHEMBL30158950

CC(C)OC(=O)c1ccc2c(c1)nc(-c1ccccn1)n2C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
CA12 O43570 1/20 0.55
CA9 Q16790 1/20 0.55
HDAC6 Q9UBN7 4/20 0.47
HDAC1 Q13547 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
JMJD6 Q6NYC1 1/20 0.46
HDAC3 O15379 2/20 0.45
HDAC2 Q92769 2/20 0.45
PADI4 Q9UM07 1/20 0.44
NAMPT P43490 1/20 0.44
CTSD P07339 3/20 0.42
FGFR1 P11362 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30158985 0.87 NPC1 (0.61) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30159104 0.84 MEN1 (0.53) NPC1RAB9AMEN1KMT2ABCAT2
SCHEMBL29876885 0.83 CA12 (0.61) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30159055 0.82 CA12 (0.47) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30158798 0.81 PADI4 (0.49) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30158779 0.76 FGFR1 (0.55) NPC1RAB9AMEN1KMT2ACA12
Trifluoroacetic Acid SCHEMBL30158966 0.76 PADI4 (0.45) NPC1RAB9AMEN1KMT2APADI4
SCHEMBL12354513 0.75 CA12 (0.66) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30159013 0.75 CA12 (0.51) NPC1RAB9AMEN1KMT2ACA12
SCHEMBL30159003 0.75 NPC1 (0.53) NPC1RAB9AMEN1KMT2ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-A Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2022-12-30 CN disclosed