SCHEMBL30176323

SCHEMBL30176323

Cc1cc(-n2c(C(C)C)c(C=O)c3cc(OCc4ccccc4)ccc32)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
S1PR3 Q99500 1/20 0.41
EDNRB P24530 2/20 0.40
EDNRA P25101 2/20 0.40
PKM P14618 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAOB P27338 3/20 0.38
MAOA P21397 2/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
LTB4R Q15722 1/20 0.37
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23886650 1.00 NPC1 (0.57) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL23898695 0.91 MEN1 (0.47) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL23898585 0.86 NPC1 (0.42) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL26654651 0.86 MEN1 (0.38) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL28995423 0.85 NPC1 (0.41) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL23886871 0.84 MEN1 (0.41) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL30176361 0.84 MEN1 (0.41) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL30176251 0.84 S1PR3 (0.44) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL23886852 0.84 S1PR3 (0.44) NPC1RAB9AMEN1KMT2AS1PR3
SCHEMBL23886916 0.84 S1PR3 (0.44) NPC1RAB9AMEN1KMT2AS1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916749-A Substituted 5-hydroxyindole compounds as alpha-1 antitrypsin modulators 弗特克斯药品有限公司 2023-04-04 CN disclosed
EP-4126817-A1 SUBSTITUTED 5-HYDROXYINDOLE COMPOUNDS AS MODULATORS OF ALPHA-1 ANTITRYPSIN Vertex Pharmaceuticals Incorporated (US) 2023-02-08 EP disclosed