SCHEMBL30183045

SCHEMBL30183045

CN(C)[C@@H]1CCN(C(=O)Cc2csc(NC(=O)c3n[nH]c4c3C(C)(C)Cc3cnc(N)nc3-4)n2)C1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F2 P00734 4/20 0.36
F10 P00742 4/20 0.36
ATR Q13535 2/20 0.34
CSNK2A1 P68400 1/20 0.33
MAPKAPK2 P49137 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21875671 1.00 F2 (0.36) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL20649089 1.00 F2 (0.36) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL21875634 1.00 F2 (0.36) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL30183507 1.00 F2 (0.36) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL30183377 0.96 F2 (0.38) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL20649013 0.96 F2 (0.38) F2F10ATRCSNK2A1MAPKAPK2
SCHEMBL21875625 0.91 F2 (0.37) F2F10ATRCSNK2A1
SCHEMBL30183032 0.91 F2 (0.37) F2F10ATRCSNK2A1
SCHEMBL21875670 0.91 F2 (0.37) F2F10ATRCSNK2A1
SCHEMBL30183504 0.91 F2 (0.37) F2F10ATRCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN claimed
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN disclosed