SCHEMBL30183263

SCHEMBL30183263

CC1(C)Cc2cnc(N)nc2-c2[nH]nc(C(=O)N3CCC(N4CCCC4)CC3)c21

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.38
L3MBTL3 Q96JM7 16/20 0.37
L3MBTL1 Q9Y468 15/20 0.37
MBTD1 Q05BQ5 4/20 0.36
TP53BP1 Q12888 2/20 0.36
L3MBTL4 Q8NA19 2/20 0.36
RAB9A P51151 1/20 0.36
ATR Q13535 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20649159 1.00 LRRK2 (0.38) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL30183348 0.99 LRRK2 (0.39) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL20649153 0.99 LRRK2 (0.39) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL20649288 0.88 ATR (0.49) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL30183353 0.88 ATR (0.49) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL20649115 0.87 ATR (0.49) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL30183153 0.87 ATR (0.49) LRRK2L3MBTL3L3MBTL1MBTD1TP53BP1
SCHEMBL20649105 0.86 ATR (0.52) LRRK2L3MBTL3L3MBTL1MBTD1L3MBTL4
SCHEMBL20649285 0.86 ATR (0.36) LRRK2L3MBTL3L3MBTL1MBTD1RAB9A
SCHEMBL30183433 0.86 ATR (0.52) LRRK2L3MBTL3L3MBTL1MBTD1L3MBTL4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN claimed
CN-110997678-B Pyrazoloquinazoline derivatives as choline kinase inhibitors 内尔维亚诺医疗科学公司 2023-02-21 CN disclosed