SCHEMBL30184050

SCHEMBL30184050

COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(N4CCN(C)C(=O)C4)c3)n[nH]c2cn1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 5/20 0.56
FGFR1 P11362 10/20 0.47
FGFR2 P21802 10/20 0.47
PIM1 P11309 2/20 0.43
KIT P10721 1/20 0.42
FLT3 P36888 1/20 0.42
FGFR4 P22455 1/20 0.41
FGFR3 P22607 1/20 0.41
NTRK1 P04629 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19949952 1.00 MAP4K1 (0.56) MAP4K1FGFR1FGFR2PIM1KIT
SCHEMBL19950352 0.94 MAP4K1 (0.60) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL19950066 0.90 MAP4K1 (0.68) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL28903704 0.90 MAP4K1 (0.51) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL19950044 0.89 MAP4K1 (0.52) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL31672290 0.89 MAP4K1 (0.52) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL19950362 0.89 MAP4K1 (0.52) MAP4K1FGFR1FGFR2PIM1KIT
SCHEMBL30183683 0.89 MAP4K1 (0.52) MAP4K1FGFR1FGFR2PIM1KIT
SCHEMBL30069603 0.88 MAP4K1 (0.60) MAP4K1FGFR1FGFR2KITFLT3
SCHEMBL19950152 0.88 MAP4K1 (0.60) MAP4K1FGFR1FGFR2KITFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4119558-A1 PYRAZOLOPYRIDINE COMPOUNDS AND USES THEREOF Incyte Corporation (US) 2023-01-18 EP claimed