SCHEMBL30187237

SCHEMBL30187237

CC(C)(C)OC(=O)N1CCN(c2nc(OCC=O)nc3c(F)c(-c4cc(O)cc5ccccc45)c(Cl)cc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 18/20 0.54
CRBN Q96SW2 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28983555 1.00 KRAS (0.54) KRASCRBNCNR1CNR2
SCHEMBL30187246 0.90 KRAS (0.51) KRASCRBN
SCHEMBL28983553 0.90 KRAS (0.51) KRASCRBN
SCHEMBL19411967 0.89 KRAS (0.61) KRAS
SCHEMBL30085115 0.89 KRAS (0.51) KRASCRBNCNR1CNR2
SCHEMBL21458461 0.89 KRAS (0.51) KRASCRBNCNR1CNR2
SCHEMBL21458459 0.89 KRAS (0.51) KRASCRBNCNR1CNR2
SCHEMBL24698376 0.87 KRAS (0.67) KRAS
SCHEMBL29125119 0.87 KRAS (0.67) KRAS
SCHEMBL30686959 0.87 KRAS (0.67) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4132655-A1 COMPOUNDS AND METHODS FOR TARGETED DEGRADATION OF KRAS Arvinas Operations, Inc. (US) 2023-02-15 EP disclosed