SCHEMBL30187752

SCHEMBL30187752

Cc1nc2sc3c(N4CC(C#N)C4)ncnc3c2c(C)c1Cl

nearest known ligand 0.98

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 13/20 0.98
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19741293 1.00 CHRM4 (0.98) CHRM4CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL30193554 0.99 CHRM4 (1.00) CHRM4CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL19741209 0.99 CHRM4 (1.00) CHRM4CYP1A2CYP3A4CYP2C9
SCHEMBL19741255 0.86 CHRM4 (0.74) CHRM4CYP1A2CYP3A4CYP2C9
SCHEMBL25711585 0.86 CHRM4 (0.74) CHRM4CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL19741358 0.85 CHRM4 (0.76) CHRM4CYP1A2CYP3A4CYP2C9
SCHEMBL30187925 0.84 CHRM4 (1.00) CHRM4CYP1A2CYP3A4CYP2C9
SCHEMBL19740788 0.84 CHRM4 (1.00) CHRM4CYP1A2CYP3A4CYP2C9
SCHEMBL19741298 0.82 CHRM4 (0.98) CHRM4CYP3A4CYP2C9
SCHEMBL30187830 0.82 CHRM4 (0.98) CHRM4CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178391-A Forward allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-05-30 CN disclosed
CN-109310668-B Positive allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-01-24 CN disclosed