SCHEMBL30187767

SCHEMBL30187767

Cc1nc2oc3c(NCC(C)C)ncnc3c2c(C)c1Cl

nearest known ligand 0.98

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 16/20 0.98
CYP1A2 P05177 1/20 0.59
KDM4E B2RXH2 3/20 0.50
MAPT P10636 1/20 0.42
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19741247 1.00 CHRM4 (0.98) CHRM4CYP1A2KDM4EMAPTUSP2
Hydrochloric Acid SCHEMBL19741379 0.99 CHRM4 (1.00) CHRM4CYP1A2KDM4EMAPTUSP2
Hydrochloric Acid SCHEMBL30193638 0.99 CHRM4 (1.00) CHRM4CYP1A2KDM4EMAPTUSP2
SCHEMBL30187885 0.87 CHRM4 (0.80) CHRM4CYP1A2KDM4EUSP2ALDH1A1
SCHEMBL19741009 0.87 CHRM4 (0.80) CHRM4CYP1A2KDM4EUSP2ALDH1A1
Hydrochloric Acid SCHEMBL19740895 0.86 CHRM4 (0.83) CHRM4CYP1A2KDM4EUSP2ALDH1A1
Hydrochloric Acid SCHEMBL30193497 0.86 CHRM4 (0.83) CHRM4CYP1A2KDM4EUSP2ALDH1A1
SCHEMBL30187701 0.85 CHRM4 (0.98) CHRM4CYP1A2KDM4EUSP2ALDH1A1
SCHEMBL19740901 0.85 CHRM4 (0.98) CHRM4CYP1A2KDM4EUSP2ALDH1A1
Hydrochloric Acid SCHEMBL19741338 0.84 CHRM4 (1.00) CHRM4CYP1A2KDM4EUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178391-A Forward allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-05-30 CN disclosed
CN-109310668-B Positive allosteric modulators of muscarinic acetylcholine receptor M4 范德比尔特大学 2023-01-24 CN disclosed