SCHEMBL30205023

SCHEMBL30205023

O=C(c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F)N1CCNCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 1.00
PARP3 Q9Y6F1 2/20 0.93
TNKS O95271 1/20 0.76
ADORA1 P30542 1/20 0.76
CDK6 Q00534 1/20 0.76
PDE3A Q14432 1/20 0.76
PARP6 Q2NL67 1/20 0.76
PARP15 Q460N3 1/20 0.76
PARP14 Q460N5 1/20 0.76
PARP10 Q53GL7 1/20 0.76
TIPARP Q7Z3E1 1/20 0.76
PARP8 Q8N3A8 1/20 0.76
PARP16 Q8N5Y8 1/20 0.76
PARP12 Q9H0J9 1/20 0.76
TNKS2 Q9H2K2 1/20 0.76
PARP11 Q9NR21 1/20 0.76
PARP2 Q9UGN5 1/20 0.76
PARP4 Q9UKK3 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL524782 1.00 PARP1 (1.00) PARP1PARP3TNKSADORA1CDK6
SCHEMBL29463415 1.00 PARP1 (1.00) PARP1PARP3TNKSADORA1CDK6
Hydrochloric Acid SCHEMBL29536089 0.99 PARP1 (0.98) PARP1PARP3TNKSADORA1CDK6
Hydrochloric Acid SCHEMBL23113141 0.99 PARP1 (0.98) PARP1PARP3TNKSADORA1CDK6
Hydrochloric Acid SCHEMBL22656793 0.99 PARP1 (0.98) PARP1PARP3TNKSADORA1CDK6
SCHEMBL864319 0.96 PARP1 (1.00) PARP1PARP3
SCHEMBL29434944 0.96 PARP1 (1.00) PARP1PARP3
SCHEMBL19569971 0.94 PARP1 (0.90) PARP1PARP3TNKSADORA1CDK6
SCHEMBL17781907 0.93 PARP1 (0.86) PARP1PARP3TNKSADORA1CDK6
SCHEMBL30293115 0.92 PARP1 (0.89) PARP1PARP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113603647-B PARP inhibitor-alkylation bifunctional molecule and preparation method and application thereof 潍坊医学院 2023-01-31 CN claimed
CN-119158026-A Compound containing PAPR1 degradation agent and BET inhibitor and application of compound in antitumor drug 成都市第三人民医院 2024-12-20 CN disclosed
CN-113603647-B PARP inhibitor-alkylation bifunctional molecule and preparation method and application thereof 潍坊医学院 2023-01-31 CN disclosed