SCHEMBL30209658

SCHEMBL30209658

O=C(Nc1ccc(C(=O)NO)cc1)Nc1ccc(-c2cccnc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.66
KDR P35968 3/20 0.62
MKNK1 Q9BUB5 3/20 0.61
MKNK2 Q9HBH9 3/20 0.61
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
NAMPT P43490 2/20 0.58
LMNA P02545 1/20 0.58
GAA P10253 1/20 0.58
CNR1 P21554 1/20 0.55
DEGS1 O15121 1/20 0.54
EPHX2 P34913 1/20 0.54
HDAC6 Q9UBN7 3/20 0.54
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28607855 1.00 HDAC1 (0.66) HDAC1KDRMKNK1MKNK2NPC1
SCHEMBL1109339 0.90 MKNK1 (0.73) HDAC1MKNK1MKNK2NPC1RAB9A
SCHEMBL28623099 0.89 KDR (0.62) HDAC1KDRNPC1RAB9ANAMPT
SCHEMBL30209636 0.89 KDR (0.62) HDAC1KDRNPC1RAB9ANAMPT
SCHEMBL28613002 0.84 HDAC1 (0.77) HDAC1GAACNR1HDAC6CYP3A4
SCHEMBL14082508 0.81 POLB (0.77) MKNK1MKNK2NPC1RAB9ANAMPT
SCHEMBL3038840 0.81 NAMPT (0.81) NPC1RAB9ANAMPTLMNAGAA
SCHEMBL14082506 0.81 NAMPT (0.86) MKNK1MKNK2NPC1RAB9ANAMPT
SCHEMBL4911349 0.81 CNR1 (0.80) KDRNPC1RAB9ANAMPTLMNA
SCHEMBL14082509 0.81 CYP11B1 (0.72) MKNK1MKNK2NPC1RAB9ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113288888-B Compounds with vasodilating activity 烟台邦杰生物科技有限公司 2023-02-03 CN claimed
CN-113288888-B Compounds with vasodilating activity 烟台邦杰生物科技有限公司 2023-02-03 CN disclosed