SCHEMBL30217007

SCHEMBL30217007

O=C(O)C1(c2cccc(Br)c2)CCS(=O)(=O)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.49
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HDAC4 P56524 3/20 0.38
HCAR3 P49019 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
FAAH O00519 1/20 0.38
TRPV1 Q8NER1 1/20 0.38
CTSD P07339 1/20 0.37
BACE1 P56817 1/20 0.37
GRK2 P25098 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29237574 1.00 AKR1C1 (0.49) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL4502888 0.87 AKR1C1 (0.65) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL671822 0.87 AKR1C1 (0.53) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL17632673 0.86 AKR1C1 (0.62) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL1492825 0.84 AKR1C1 (0.59) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL22832447 0.81 AKR1C1 (0.43) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL30967898 0.80 AKR1C1 (0.46) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL11832779 0.80 AKR1C1 (0.46) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL14332444 0.80 AKT1 (0.46) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1
SCHEMBL29237470 0.80 AKR1C1 (0.46) AKR1C1ALDH1A1GAASMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4396179-A1 INDOLE COMPOUNDS AND METHODS OF USE GENZYME CORPORATION (US) 2024-07-10 EP disclosed
CN-118201919-A Indole compounds and methods of use 健赞公司 2024-06-14 CN disclosed
WO-2023034992-A1 INDOLE COMPOUNDS AND METHODS OF USE GENZYME CORPORATION (US) 2023-03-09 WO disclosed