SCHEMBL30220149

SCHEMBL30220149

CCCCOc1nc(N)c2cnn(Cc3ccc(CN4CCCC4)cc3)c2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 1.00
CYP2D6 P10635 4/20 0.98
TLR7 Q9NYK1 13/20 0.55
IL6 P05231 1/20 0.51
TSHR P16473 1/20 0.50
TLR8 Q9NR97 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20210107 1.00 CYP3A4 (1.00) CYP3A4CYP2D6TLR7IL6TSHR
SCHEMBL20210102 0.99 CYP3A4 (1.00) CYP3A4CYP2D6TLR7IL6TSHR
Hydrochloric Acid SCHEMBL23234423 0.99 CYP3A4 (0.98) CYP3A4CYP2D6TLR7IL6TSHR
Hydrochloric Acid SCHEMBL23234422 0.99 CYP3A4 (0.98) CYP3A4CYP2D6TLR7IL6TSHR
SCHEMBL20210101 0.98 CYP3A4 (1.00) CYP3A4CYP2D6TLR7IL6TSHR
SCHEMBL20210108 0.92 CYP3A4 (1.00) CYP3A4CYP2D6TLR7IL6TLR8
SCHEMBL21482063 0.91 CYP3A4 (0.84) CYP3A4CYP2D6TLR7IL6
SCHEMBL20209845 0.91 CYP3A4 (1.00) CYP3A4CYP2D6TLR7IL6TLR8
SCHEMBL20209842 0.90 CYP3A4 (0.96) CYP3A4CYP2D6TLR7IL6TLR8
SCHEMBL20209833 0.90 CYP3A4 (0.81) CYP3A4CYP2D6TLR7TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513039-B TLR7 agonist prodrug, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-01-24 CN disclosed