SCHEMBL30224397

SCHEMBL30224397

FC(F)(F)Cn1nc(C(F)(F)F)c2ccc(Br)cc21

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.44
NT5E P21589 1/20 0.35
SSTR4 P31391 1/20 0.34
KDM4C Q9H3R0 2/20 0.34
SLC2A1 P11166 1/20 0.33
SLC2A3 P11169 1/20 0.33
PDGFRA P16234 1/20 0.33
CDK5 Q00535 1/20 0.33
TYRO3 Q06418 1/20 0.33
RORC P51449 2/20 0.32
LMNA P02545 1/20 0.32
KMO O15229 1/20 0.31
AKR1B1 P15121 2/20 0.31
AKR1A1 P14550 1/20 0.31
DGAT1 O75907 1/20 0.31
MAPT P10636 1/20 0.31
CCR1 P32246 1/20 0.31
CYP11B2 P19099 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23994535 1.00 ESR1 (0.44) ESR1NT5ESSTR4KDM4CSLC2A1
SCHEMBL30224393 1.00 ESR1 (0.44) ESR1NT5ESSTR4KDM4CSLC2A1
SCHEMBL22152000 0.84 PDGFRA (0.34) ESR1NT5ESSTR4SLC2A1SLC2A3
SCHEMBL23993249 0.83 ESR1 (0.45) ESR1KDM4CPDGFRACDK5TYRO3
SCHEMBL30224924 0.83 ESR1 (0.45) ESR1KDM4CPDGFRACDK5TYRO3
SCHEMBL23993327 0.82 ESR1 (0.44) ESR1NT5EKDM4CPDGFRACDK5
SCHEMBL31636216 0.82 PDGFRA (0.48) ESR1KDM4CPDGFRACDK5TYRO3
SCHEMBL1965696 0.80 ESR1 (0.43) ESR1KDM4CPDGFRACDK5TYRO3
SCHEMBL23993144 0.78 ESR1 (0.41) ESR1KDM4CPDGFRACDK5TYRO3
SCHEMBL23993488 0.78 ESR1 (0.41) ESR1KDM4CPDGFRACDK5TYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143194-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-03-08 EP disclosed