SCHEMBL30239885

SCHEMBL30239885

NCCNc1nonc1C(=Nc1ccc(F)c(Br)c1)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 20/20 1.00
CYP3A4 P08684 1/20 0.76
CYP2C9 P11712 1/20 0.76
TDO2 P48775 1/20 0.76
IDO2 Q6ZQW0 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL149285 0.87 IDO1 (1.00) IDO1TDO2IDO2
Epacadostat SCHEMBL30521952 0.87 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
Epacadostat SCHEMBL145947 0.87 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
Epacadostat SCHEMBL148867 0.87 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
Epacadostat SCHEMBL19808101 0.87 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
SCHEMBL144582 0.85 IDO1 (0.89) IDO1CYP3A4CYP2C9TDO2IDO2
SCHEMBL145813 0.85 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
SCHEMBL2512595 0.84 IDO1 (1.00) IDO1CYP3A4CYP2C9TDO2IDO2
SCHEMBL2521517 0.84 IDO1 (1.00) IDO1
SCHEMBL144215 0.83 IDO1 (0.89) IDO1CYP3A4CYP2C9TDO2IDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113527368-B Preparation method and application of compound and anti-cancer drug 中国科学技术大学 2023-03-10 CN disclosed
WO-2023015526-A1 COMPOUND, PREPARATION METHOD FOR ANTI-CANCER DRUG, AND USE 中国科学技术大学 2023-02-16 WO disclosed