SCHEMBL30252552

SCHEMBL30252552

Nc1cc(-c2nccs2)nc(-c2cc(Cl)cc(Br)n2)c1Br

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
CYP1A1 P04798 4/20 0.39
CYP1A2 P05177 4/20 0.39
CYP1B1 Q16678 4/20 0.39
HSP90AA1 P07900 1/20 0.38
ADORA1 P30542 3/20 0.32
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30252564 0.85 ADORA2A (0.41) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL20911562 0.85 ADORA2A (0.41) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30252375 0.82 ADORA2A (0.58) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL20911255 0.82 ADORA2A (0.58) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30253171 0.82 CYP1A1 (0.42) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30252648 0.81 ADORA2A (0.40) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL20911213 0.81 ADORA2A (0.42) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30252710 0.81 ADORA2A (0.42) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30253003 0.81 ADORA2A (0.39) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1
SCHEMBL30252999 0.80 ADORA2A (0.41) ADORA2ACYP1A1CYP1A2CYP1B1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed