SCHEMBL30257537

SCHEMBL30257537

Cn1nc(C2CC2)cc1Oc1cc(C#N)ccc1-c1ncc(CCN)cn1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
AXL P30530 1/20 0.34
TYRO3 Q06418 1/20 0.34
MERTK Q12866 1/20 0.34
KDM1A O60341 2/20 0.32
NSD2 O96028 2/20 0.32
ALOX5AP P20292 4/20 0.31
FEN1 P39748 4/20 0.31
SCN9A Q15858 3/20 0.31
PTH1R Q03431 2/20 0.31
GPR119 Q8TDV5 1/20 0.31
GRM5 P41594 2/20 0.31
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554329 1.00 CYP19A1 (0.34) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL30257409 0.96 FEN1 (0.35) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25554245 0.96 FEN1 (0.35) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25554463 0.96 PTH1R (0.35) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25058332 0.94 PDE2A (0.34) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL30353054 0.93 NSD2 (0.35) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25554344 0.93 NSD2 (0.35) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25554675 0.91 LRRK2 (0.34) CYP19A1CYP11B1CYP11B2
SCHEMBL30257448 0.90 KDM1A (0.36) CYP19A1CYP11B1CYP11B2AXLTYRO3
SCHEMBL25554123 0.90 KDM1A (0.36) CYP19A1CYP11B1CYP11B2AXLTYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed
EP-4137481-A1 ARYL OR HETEROARYL DERIVATIVE Teijin Pharma Limited (JP) 2023-02-22 EP disclosed