SCHEMBL30270446

SCHEMBL30270446

O=S(=O)(Cl)N1CCC(c2cccnc2F)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.41
COMT P21964 2/20 0.39
SPR P35270 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
HTR2B P41595 2/20 0.36
CHRM5 P08912 2/20 0.35
TP53 P04637 1/20 0.35
HTR2A P28223 1/20 0.35
HTR6 P50406 1/20 0.35
HTR1A P08908 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26213657 1.00 HCAR2 (0.41) HCAR2COMTSPRPTGDR2HTR2B
SCHEMBL30269813 0.88 COMT (0.41) HCAR2COMTSPRPTGDR2HTR2B
SCHEMBL26213669 0.81 HCAR2 (0.37) HCAR2COMTSPRPTGDR2
SCHEMBL32162354 0.79 HCAR2 (0.48) HCAR2HTR1ASLC6A2SLC6A4
SCHEMBL2460605 0.79 HCAR2 (0.48) HCAR2HTR1ASLC6A2SLC6A4
SCHEMBL26214485 0.79 KIT (0.40) HCAR2COMTSPRPTGDR2
SCHEMBL23235688 0.77 HCAR2 (0.47) HCAR2SPR
SCHEMBL13361555 0.76 HCAR2 (0.46) HCAR2HTR1ASLC6A2SLC6A4
SCHEMBL3319484 0.75 KDM4E (0.48) SPR
SCHEMBL7710106 0.74 HCAR2 (0.44) HCAR2SPRHTR1ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115843271-B Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2024-08-13 CN disclosed
CN-115843271-A Indole derivatives and their use for the treatment of cancer 克洛德贝纳尔-里昂第一大学 2023-03-24 CN disclosed