SCHEMBL30273129

SCHEMBL30273129

Clc1cc(N2CCOCC2)nc(OCCc2ccccn2)n1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 2/20 0.72
SYK P43405 2/20 0.72
IRAK4 Q9NWZ3 2/20 0.72
BRSK1 Q8TDC3 1/20 0.72
FES P07332 1/20 0.58
FER P16591 1/20 0.58
FRK P42685 1/20 0.58
CAMK1D Q8IU85 1/20 0.58
PIKFYVE Q9Y2I7 1/20 0.58
PIK3CA P42336 10/20 0.55
PIK3CB P42338 2/20 0.46
PIK3CG P48736 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
FFAR1 O14842 1/20 0.46
KMT2A Q03164 2/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1617807 1.00 TYK2 (0.72) TYK2SYKIRAK4BRSK1FES
SCHEMBL3560513 0.90 PIK3CA (0.66) TYK2SYKIRAK4BRSK1FES
SCHEMBL11929833 0.86 TYK2 (0.72) TYK2SYKIRAK4BRSK1FES
SCHEMBL3110596 0.86 TYK2 (0.75) TYK2SYKIRAK4BRSK1FES
SCHEMBL12634088 0.85 TYK2 (0.70) TYK2SYKIRAK4BRSK1FES
SCHEMBL1877075 0.84 TYK2 (0.68) TYK2SYKIRAK4BRSK1FES
SCHEMBL31025329 0.84 TYK2 (1.00) TYK2SYKIRAK4BRSK1FES
SCHEMBL1616481 0.84 TYK2 (1.00) TYK2SYKIRAK4BRSK1FES
SCHEMBL30273130 0.84 TYK2 (1.00) TYK2SYKIRAK4BRSK1FES
SCHEMBL1617732 0.83 TYK2 (0.61) TYK2SYKIRAK4BRSK1FES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113683596-B Pyrimidine tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2023-02-10 CN claimed
CN-113683596-B Pyrimidine tankyrase 2 inhibitor and preparation method and application thereof 上海应用技术大学 2023-02-10 CN disclosed