SCHEMBL30273142

SCHEMBL30273142

O=c1[nH]c2cc(CCl)ccc2c2cscc12

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.43
KIF11 P52732 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.33
TNKS O95271 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
GPR3 P46089 1/20 0.33
BLM P54132 1/20 0.33
PMP22 Q01453 1/20 0.33
KMT2A Q03164 1/20 0.33
PARP15 Q460N3 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30273140 0.84 PARP1 (0.61) PARP1KIF11KDM4EALDH1A1
SCHEMBL7027018 0.77 PARP1 (0.48) PARP1KIF11KDM4EALDH1A1
SCHEMBL30577720 0.76 PARP1 (0.74) PARP1KDM4EPARP15TNKS2
SCHEMBL13688018 0.76 PARP1 (0.69) PARP1KIF11KDM4EALDH1A1MEN1
SCHEMBL25093568 0.73 PARP1 (0.46) PARP1KDM4EALDH1A1
SCHEMBL30577714 0.73 PARP1 (0.46) PARP1KDM4EALDH1A1
SCHEMBL25738485 0.72 PARP1 (0.38) PARP1KIF11KDM4EALDH1A1LMNA
SCHEMBL29203560 0.72 PARP1 (0.68) PARP1KIF11KDM4EALDH1A1KMT2A
SCHEMBL10134731 0.72 FLT3 (0.44) PARP1
SCHEMBL25093566 0.71 PARP1 (0.51) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240368169-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS (SHANGHAI), INC. (CN) 2024-11-07 US disclosed
EP-4392425-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF Impact Therapeutics (Shanghai), Inc. (CN) 2024-07-03 EP disclosed
WO-2023025307-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF IMPACT THERAPEUTICS (SHANGHAI) , INC (CN) 2023-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240368169-A1 SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF PARP1, PARP2, PARP11 PARP1 1/4885KIF11 3787/4885KDM4E 2747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.