SCHEMBL30289264

SCHEMBL30289264

Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(CN3CCC(NC(=O)OC(C)(C)C)CC3)cc21

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 8/20 0.57
CRBN Q96SW2 8/20 0.57
PARP1 P09874 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
AKT1 P31749 1/20 0.40
DRD2 P14416 3/20 0.40
KCNA3 P22001 1/20 0.40
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
PRKDC P78527 1/20 0.39
MCHR1 Q99705 2/20 0.38
NSD2 O96028 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30289493 0.98 DDB1 (0.55) DDB1CRBNPARP1PARP2AKT1
SCHEMBL30289081 0.97 DDB1 (0.54) DDB1CRBNPARP1PARP2AKT1
SCHEMBL30289475 0.93 DDB1 (0.56) DDB1CRBNPARP1PARP2DRD2
SCHEMBL26099950 0.91 DDB1 (0.52) DDB1CRBNPARP1PARP2AKT1
SCHEMBL26100681 0.91 DDB1 (0.52) DDB1CRBNPARP1PARP2AKT1
SCHEMBL23832582 0.91 CRBN (0.49) DDB1CRBNPARP1PARP2AKT1
SCHEMBL30289386 0.91 DDB1 (0.54) DDB1CRBNPARP1PARP2DRD2
SCHEMBL26102788 0.90 DDB1 (0.51) DDB1CRBNPARP1PARP2AKT1
SCHEMBL26098410 0.90 DDB1 (0.51) DDB1CRBNPARP1PARP2AKT1
SCHEMBL21070822 0.90 CRBN (0.51) DDB1CRBNPARP1PARP2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4405359-A2 MDM2 DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2024-07-31 EP disclosed
WO-2023049790-A2 MDM2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2023-03-30 WO disclosed