SCHEMBL30295752

SCHEMBL30295752

Cc1nc(N2CCC3(CC2)CO[C@@H](C)[C@H]3N)c(CO)nc1Sc1ccnc(N2CC3(COC3)C2)c1Cl

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.79
KCNH2 Q12809 2/20 0.56
EGFR P00533 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26981001 1.00 PTPN11 (0.79) PTPN11KCNH2EGFR
SCHEMBL21115042 1.00 PTPN11 (0.79) PTPN11KCNH2EGFR
SCHEMBL21154416 0.95 PTPN11 (0.76) PTPN11KCNH2EGFR
SCHEMBL19785589 0.92 PTPN11 (0.81) PTPN11KCNH2EGFR
SCHEMBL30295728 0.92 PTPN11 (0.81) PTPN11KCNH2EGFR
SCHEMBL19785614 0.90 PTPN11 (0.80) PTPN11KCNH2EGFR
SCHEMBL30295924 0.90 PTPN11 (0.80) PTPN11KCNH2EGFR
SCHEMBL25261253 0.90 PTPN11 (0.75) PTPN11KCNH2EGFR
SCHEMBL21154584 0.89 PTPN11 (0.86) PTPN11KCNH2EGFR
SCHEMBL21115105 0.89 PTPN11 (0.73) PTPN11KCNH2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478131-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-116478132-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-109983001-B 2, 5-disubstituted 3-methylpyrazines and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-04-04 CN disclosed