SCHEMBL30296136

SCHEMBL30296136

Cc1nc(N2CCC(C)(N)CC2)cnc1-c1ccccc1Cl

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.65
KCNH2 Q12809 5/20 0.65
MAPK3 P27361 3/20 0.65
MAPK1 P28482 3/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19785336 1.00 PTPN11 (0.65) PTPN11KCNH2MAPK3MAPK1
SCHEMBL30295870 0.91 PTPN11 (0.80) PTPN11KCNH2MAPK3MAPK1
SCHEMBL19785300 0.91 PTPN11 (0.80) PTPN11KCNH2MAPK3MAPK1
SCHEMBL25514349 0.90 PTPN11 (0.53) PTPN11KCNH2MAPK3MAPK1
SCHEMBL23425127 0.86 PTPN11 (0.50) PTPN11KCNH2MAPK3MAPK1
SCHEMBL30296115 0.86 PTPN11 (0.65) PTPN11KCNH2MAPK3MAPK1
SCHEMBL19785338 0.86 PTPN11 (0.65) PTPN11KCNH2MAPK3MAPK1
SCHEMBL21154819 0.83 PTPN11 (0.54) PTPN11KCNH2MAPK3MAPK1
SCHEMBL24233637 0.82 PTPN11 (0.52) PTPN11KCNH2MAPK3MAPK1
SCHEMBL30296123 0.81 PTPN11 (0.80) PTPN11KCNH2MAPK3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478131-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-116478132-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-109983001-B 2, 5-disubstituted 3-methylpyrazines and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-04-04 CN disclosed