SCHEMBL30296997

SCHEMBL30296997

COc1ccc(C#CC2c3ccccc3CCN2c2cccc(OC)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 6/20 0.50
KMT2A Q03164 2/20 0.43
GAA P10253 1/20 0.43
GFER P55789 1/20 0.43
DRD2 P14416 4/20 0.42
DRD5 P21918 4/20 0.42
DRD3 P35462 3/20 0.42
DRD4 P21917 3/20 0.42
GID4 Q8IVV7 2/20 0.41
GRIN2B Q13224 1/20 0.40
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29170190 1.00 DRD1 (0.50) DRD1KMT2AGAAGFERDRD2
SCHEMBL30296985 0.92 DRD1 (0.44) DRD1KMT2AGAAGFERDRD2
SCHEMBL30297017 0.91 DRD1 (0.44) DRD1KMT2AGAAGFERMEN1
SCHEMBL29170205 0.91 DRD1 (0.45) DRD1KMT2AGAADRD2DRD5
SCHEMBL30296945 0.91 DRD1 (0.45) DRD1KMT2AGAADRD2DRD5
SCHEMBL30296994 0.86 DRD1 (0.42) DRD1KMT2ADRD2DRD5DRD3
SCHEMBL30296909 0.85 DRD1 (0.41) DRD1KMT2ADRD2DRD5DRD3
SCHEMBL30297007 0.85 DRD1 (0.41) DRD1KMT2ADRD2DRD4GID4
SCHEMBL29170196 0.85 DRD1 (0.41) DRD1KMT2ADRD2DRD5DRD3
SCHEMBL28615700 0.79 ESR1 (0.39) GAAGFERGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117384094-A Preparation method of alkynyl tetrahydroisoquinoline derivative 江苏中利集团股份有限公司 2024-01-12 CN disclosed
CN-115894364-A Preparation method of alkynyl tetrahydroisoquinoline derivatives 江苏中利集团股份有限公司 2023-04-04 CN disclosed