SCHEMBL30353065

SCHEMBL30353065

Cn1nc(-c2cccc(F)c2)cc1Oc1cc(C#N)ccc1-c1ncc(CCN)cn1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.39
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
CYP19A1 P11511 2/20 0.36
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRA3 P34903 3/20 0.36
GABRA5 P31644 2/20 0.36
TAAR1 Q96RJ0 1/20 0.34
SCN9A Q15858 1/20 0.34
ICMT O60725 2/20 0.34
ADRA2C P18825 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
MET P08581 1/20 0.34
NSD2 O96028 1/20 0.33
PTGER1 P34995 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554479 1.00 GRM5 (0.39) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL25554247 0.92 CYP11B1 (0.41) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL25554119 0.92 GRM5 (0.38) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL30353104 0.92 GRM5 (0.38) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL30256876 0.90 TAAR1 (0.42) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL25554091 0.90 TAAR1 (0.42) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL25554092 0.87 GRM5 (0.41) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL30257088 0.87 GRM5 (0.41) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL25251491 0.87 GRM5 (0.38) GRM5CYP11B1CYP11B2CYP19A1GABRG2
SCHEMBL30257430 0.87 GRM5 (0.38) GRM5CYP11B1CYP11B2CYP19A1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed