SCHEMBL30366702

SCHEMBL30366702

Cc1cccc(Oc2ccc(-c3c(C4=CCNCC4)n(C)c4c(C#N)cnc(N)c34)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.39
FFAR4 Q5NUL3 1/20 0.31
PIK3CD O00329 1/20 0.31
CCNT1 O60563 1/20 0.31
CDK9 P50750 1/20 0.31
KDR P35968 2/20 0.30
TEK Q02763 2/20 0.30
LCK P06239 1/20 0.30
PRMT5 O14744 3/20 0.30
ATR Q13535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28981099 0.84 BTK (0.39) BTKFFAR4KDRTEKLCK
SCHEMBL30366701 0.81 BTK (0.36) BTKFFAR4
SCHEMBL30366769 0.80 KDR (0.35) FFAR4KDRTEKLCK
SCHEMBL30366523 0.77 KDR (0.33) FFAR4KDRTEKLCK
SCHEMBL28981103 0.76 BTK (0.35) BTKPRMT5
SCHEMBL30325807 0.76 BTK (0.40) BTK
SCHEMBL30366804 0.76 CYP3A4 (0.47) BTKFFAR4KDRTEK
SCHEMBL30366502 0.75 CYP3A4 (0.42) BTKFFAR4KDRTEK
SCHEMBL31411040 0.75 LCK (0.41) BTKKDRTEKLCK
SCHEMBL22678110 0.75 LCK (0.41) BTKKDRTEKLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed