SCHEMBL30367484

SCHEMBL30367484

CCn1nc(N2C(=O)c3ccccc3C2=O)c2c(I)cc(Br)cc21

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 2/20 0.36
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
MAPK1 P28482 1/20 0.31
GSK3B P49841 1/20 0.31
BRD1 O95696 2/20 0.31
TAF1 P21675 2/20 0.31
BRPF1 P55201 2/20 0.31
HTR3A P46098 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA2B P29275 1/20 0.30
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30367868 0.84 MAPK13 (0.35) CYP1B1KMT2AMEN1RAB9AMAPK1
SCHEMBL30367512 0.70 MAPK1 (0.38) KMT2AMEN1MAPK1GSK3B
SCHEMBL31052465 0.69 KDM4E (0.40) KMT2AMEN1GAAMAPK1
SCHEMBL419865 0.68 KDR (0.35) NR1H2NR1H3KMT2AMEN1RAB9A
SCHEMBL10112088 0.65 DNMT1 (0.40) NR1H2NR1H3KMT2AMEN1GAA
SCHEMBL31439960 0.65 MEN1 (0.38) NR1H2NR1H3KMT2AMEN1GAA
SCHEMBL423584 0.64 KDR (0.41) KMT2AMEN1
SCHEMBL420191 0.63 NR1H3 (0.40) NR1H3KMT2AMEN1GAAMAPK1
SCHEMBL21114112 0.62 ADORA2A (0.43) NR1H2NR1H3GAAADORA2AADORA2B
SCHEMBL30274181 0.62 ADORA2A (0.43) NR1H2NR1H3GAAADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023155886-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-08-24 WO disclosed
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed
WO-2023051464-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-04-06 WO disclosed